SCHEMBL8322935

SCHEMBL8322935

COC(=O)c1ccc(CCc2cc(Br)ccc2OCc2ccccc2)cc1O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.49
ALDH1A1 P00352 2/20 0.48
USP28 Q96RU2 1/20 0.48
USP25 Q9UHP3 1/20 0.48
RAB9A P51151 1/20 0.48
LMNA P02545 4/20 0.47
HTT P42858 2/20 0.47
PTGER1 P34995 5/20 0.46
LRRK2 Q5S007 2/20 0.46
CYP1A2 P05177 1/20 0.46
USP2 O75604 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8325136 0.90 ABCB1 (0.51) CCR5ALDH1A1USP28USP25RAB9A
SCHEMBL8321056 0.89 FOLH1 (0.51) CCR5ALDH1A1USP28USP25RAB9A
SCHEMBL8321603 0.88 PTGER1 (0.54) LMNAPTGER1LRRK2HPGD
SCHEMBL8319729 0.88 ABCB1 (0.56) LMNAPTGER1HPGD
SCHEMBL8324955 0.88 MTNR1A (0.59)
SCHEMBL8327489 0.85 LMNA (0.43) LMNAHTTPTGER1HPGD
SCHEMBL8324940 0.85 CCR5 (0.53) CCR5ALDH1A1USP28USP25RAB9A
SCHEMBL8409537 0.85 CCR5 (0.53) CCR5ALDH1A1USP28USP25RAB9A
SCHEMBL8324067 0.83 ABCB1 (0.53) CCR5PTGER1LRRK2CYP1A2
SCHEMBL8324057 0.82 PTGER4 (0.59) LMNAPTGER1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed