SCHEMBL8325136

SCHEMBL8325136

COC(=O)c1ccc(CCc2cc(Br)ccc2OCc2ccccc2)cc1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.51
ABCG2 Q9UNQ0 1/20 0.51
MTNR1A P48039 2/20 0.50
MTNR1B P49286 2/20 0.50
CCR5 P51681 2/20 0.49
LRRK2 Q5S007 1/20 0.48
USP28 Q96RU2 1/20 0.48
USP25 Q9UHP3 1/20 0.48
ALDH1A1 P00352 1/20 0.48
RAB9A P51151 1/20 0.48
LMNA P02545 2/20 0.47
APP P05067 1/20 0.47
HTT P42858 1/20 0.47
HDAC1 Q13547 2/20 0.47
SMPD1 P17405 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC2 Q92769 1/20 0.46
CYP1A2 P05177 1/20 0.46
PTGER1 P34995 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8324067 0.92 ABCB1 (0.53) ABCB1ABCG2MTNR1AMTNR1BCCR5
SCHEMBL8322935 0.90 CCR5 (0.49) CCR5LRRK2USP28USP25ALDH1A1
SCHEMBL8325289 0.88 ABCB1 (0.62) ABCB1ABCG2MTNR1AMTNR1BLMNA
SCHEMBL8324940 0.85 CCR5 (0.53) ABCB1ABCG2CCR5USP28USP25
SCHEMBL8409537 0.85 CCR5 (0.53) ABCB1ABCG2CCR5USP28USP25
SCHEMBL8326037 0.82 CCR5 (0.46) MTNR1AMTNR1BCCR5LRRK2USP28
SCHEMBL14891403 0.82 FFAR4 (0.54) CCR5LRRK2ALDH1A1LMNAHDAC1
SCHEMBL8322308 0.82 PTGER4 (0.59) ABCB1ABCG2MTNR1AMTNR1BLMNA
SCHEMBL8323808 0.81 CCR5 (0.47) MTNR1AMTNR1BCCR5LRRK2USP28
SCHEMBL8321056 0.81 FOLH1 (0.51) CCR5USP28USP25ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733033-B1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LTD (GB) 1999-12-22 EP disclosed
US-5811459-A PAIN RELIEVERS ZENECA LIMITED (GB) 1998-09-22 US disclosed
EP-0733033-A1 PHARMACEUTICALLY ACTIVE SUBSTITUTED AROMATIC COMPOUNDS ZENECA LIMITED (GB) 1996-09-25 EP disclosed