SCHEMBL8327484

SCHEMBL8327484

[CH2]CC(C)(c1ccccc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.40
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
PLA2G1B P04054 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
CYP19A1 P11511 1/20 0.33
HTT P42858 1/20 0.33
PTGS2 P35354 1/20 0.33
KCNN4 O15554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328588 0.80 KIF11 (0.45) KIF11CNR1CNR2CYP19A1TSHR
SCHEMBL8326409 0.79 KIF11 (0.44) KIF11NPC1RAB9ACYP3A4CYP2D6
SCHEMBL8320416 0.79 KIF11 (0.44) KIF11NPC1RAB9ACYP3A4CYP2D6
SCHEMBL8325626 0.78 KCNN4 (0.43) KIF11CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4249887 0.77 TAAR1 (0.46) CYP3A4CYP2D6CYP2C9CYP2C19KCNN4
SCHEMBL8329053 0.74 ALDH1A1 (0.56) KIF11NPC1RAB9ACYP3A4CYP2D6
SCHEMBL8324979 0.73 TSHR (0.45) KIF11RAB9ACYP3A4CYP2D6CYP1A2
SCHEMBL8325767 0.72 KIF11 (0.46) KIF11CYP3A4TSHR
SCHEMBL530151 0.72 HTT (0.42) KIF11RAB9ACYP2C19HTTAKR1C3
SCHEMBL8324574 0.71 KIF11 (0.46) KIF11CYP3A4CYP2D6KCNH2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed