SCHEMBL8326409

SCHEMBL8326409

[CH2]CC(N)(c1ccccc1)c1ccc(F)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.44
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KCNN4 O15554 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
PLA2G1B P04054 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ATG4B Q9Y4P1 1/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
PHOSPHO1 Q8TCT1 1/20 0.35
CYP19A1 P11511 1/20 0.34
SLC6A2 P23975 1/20 0.33
KCNH2 Q12809 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8320416 1.00 KIF11 (0.44) KIF11NPC1RAB9AKCNN4CYP3A4
SCHEMBL8324065 0.80 KIF11 (0.50) KIF11KCNN4CYP19A1
SCHEMBL8327484 0.79 KIF11 (0.40) KIF11NPC1RAB9AKCNN4CYP3A4
SCHEMBL8327109 0.77 KCNN4 (0.48) KIF11KCNN4
SCHEMBL8326422 0.77 KCNN4 (0.48) KIF11KCNN4
SCHEMBL27525548 0.76 KCNN4 (0.52) KIF11KCNN4CYP2D6CYP1A2CYP2C9
SCHEMBL8321948 0.76 KIF11 (0.49) KIF11KCNN4
SCHEMBL8321573 0.76 KIF11 (0.49) KIF11KCNN4
SCHEMBL8321366 0.73 ALDH1A1 (0.58) KIF11KCNN4SLC6A4SLC6A3CYP19A1
SCHEMBL8322782 0.73 ALDH1A1 (0.58) KIF11KCNN4SLC6A4SLC6A3CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948496-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDONE COMPOUNDS AND METHODS OF USE Amgen inc. (US) 1999-10-13 EP disclosed
WO-1998024780-A2 SUBSTITUTED PYRIMIDINONE AND PYRIDINONE COMPOUNDS AND THEIR USE AMGEN INC. (US) 1998-06-11 WO disclosed