SCHEMBL8330647

SCHEMBL8330647

O=C1Nc2c(ccc3c2CN(Cc2ccccc2)C3)C1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 2/20 0.43
PTGS2 P35354 1/20 0.43
ACHE P22303 2/20 0.42
PNMT P11086 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
GAA P10253 1/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
MAPT P10636 2/20 0.38
MAPK1 P28482 2/20 0.38
TP53 P04637 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP1A2 P05177 1/20 0.38
CES1 P23141 2/20 0.38
NSD2 O96028 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330468 0.84 MEN1 (0.38) BCHEPTGS2ACHEPNMTGAA
SCHEMBL8330462 0.84 MEN1 (0.38) BCHEPTGS2ACHEPNMTGAA
SCHEMBL8329206 0.81 CES1 (0.40) BCHEPNMTALDH1A1LMNAMAPT
SCHEMBL3842915 0.73 SLC6A5 (0.46) ACHEDRD2SLC6A5
SCHEMBL8327753 0.73 CES1 (0.42) BCHEALDH1A1KDM4ECES1NSD2
SCHEMBL8331316 0.70 CES1 (0.40) BCHEALDH1A1CES1NSD2DAO
SCHEMBL8331051 0.70 CES1 (0.40) BCHEALDH1A1CES1NSD2DAO
SCHEMBL1671165 0.68 EPHX2 (0.56) ACHEGAAALDH1A1KMT2ASIGMAR1
SCHEMBL8450698 0.68 SIGMAR1 (0.58) ACHEPNMTALDH1A1LMNACYP1A2
SCHEMBL6672942 0.67 SIGMAR1 (0.62) ACHELMNACYP1A2SIGMAR1HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed