SCHEMBL8329239

SCHEMBL8329239

CN1Cc2c(Cl)cc3c(c2C1)NC(=O)C3=O

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES1 P23141 11/20 0.47
DNMT1 P26358 1/20 0.47
DAO P14920 2/20 0.40
NSD2 O96028 1/20 0.40
BCHE P06276 1/20 0.40
ALDH1A1 P00352 1/20 0.38
ALDH2 P05091 1/20 0.38
ALDH3A1 P30838 1/20 0.38
TGM2 P21980 2/20 0.37
CASP7 P55210 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CASP3 P42574 2/20 0.31
CASP1 P29466 1/20 0.31
CASP9 P55211 1/20 0.31
CA7 P43166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331553 0.81 ALDH1A1 (0.49) CES1DNMT1DAONSD2BCHE
SCHEMBL6609048 0.77 MAOA (0.40) CES1DAONSD2BCHEALDH1A1
SCHEMBL13232796 0.74 CES1 (0.36) CES1DNMT1ALDH1A1ALDH2ALDH3A1
SCHEMBL4350619 0.74 ALDH1A1 (0.44) CES1DNMT1BCHEALDH1A1ALDH2
SCHEMBL8102934 0.74 CES1 (0.39) CES1DNMT1ALDH1A1TGM2
SCHEMBL8327753 0.73 CES1 (0.42) CES1DAONSD2BCHEALDH1A1
SCHEMBL6607897 0.70 CYP2C9 (0.39) ALDH1A1
SCHEMBL6609831 0.68 MCHR1 (0.39) TGM2
SCHEMBL13592440 0.68 GRIA1 (0.36) CES1ALDH1A1ALDH2ALDH3A1L3MBTL1
SCHEMBL24690819 0.68 CES1 (0.61) CES1DNMT1DAONSD2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed