SCHEMBL8328137

SCHEMBL8328137

CCCc1cc(C)cc(-n2c(C)ccc2C)n1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 6/20 0.51
NOS1 P29475 4/20 0.51
NOS3 P29474 3/20 0.51
MAPT P10636 2/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.36
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
SREBF2 Q12772 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326929 0.86 NOS2 (0.48) NOS2NOS1NOS3KDM4EALDH1A1
SCHEMBL13040665 0.85 NOS2 (0.42) NOS2NOS1NOS3
SCHEMBL2834751 0.85 NOS1 (0.44) NOS2NOS1NOS3
SCHEMBL5672155 0.85 NOS2 (0.36) NOS2NOS1NOS3
SCHEMBL8329772 0.85 NOS2 (0.39) NOS2NOS1NOS3
SCHEMBL2830408 0.83 NOS1 (0.57) NOS2NOS1NOS3
SCHEMBL13040656 0.82 NOS2 (0.55) NOS2NOS1NOS3
SCHEMBL8329387 0.82 NOS2 (0.55) NOS2NOS1NOS3
SCHEMBL8330516 0.81 NOS2 (0.33) NOS2NOS1NOS3
SCHEMBL8330518 0.81 NOS2 (0.40) NOS2NOS1NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8932842-B2 Aminopyridine dimer compounds, compositions and related methods for neuronal nitric oxide synthase inhibition NORTHWESTERN UNIVERSITY (US) 2015-01-13 US disclosed
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
US-5962442-A ADMINISTERING A 3-OXO-4-AZASTEROID MERCK & CO., INC. (US) 1999-10-05 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed