SCHEMBL8328262

SCHEMBL8328262

CC(C)(C)OC(=O)N(Cc1ccc(F)cc1)CC(O)COC(=O)C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC2 Q92769 1/20 0.40
NCOR2 Q9Y618 1/20 0.40
ADRB2 P07550 2/20 0.39
ADRB1 P08588 2/20 0.39
ADRB3 P13945 2/20 0.39
KCNQ4 P56696 3/20 0.37
KCNQ5 Q9NR82 3/20 0.37
BACE1 P56817 3/20 0.37
RIPK1 Q13546 2/20 0.36
KDM1A O60341 2/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
ABCB1 P08183 2/20 0.35
NR1D1 P20393 1/20 0.35
GRM2 Q14416 1/20 0.35
NPC1 O15118 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328009 0.88 ADRB2 (0.44) ADRB2ADRB1ADRB3RIPK1ABCB1
SCHEMBL8323152 0.87 KDM1A (0.37) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL8327226 0.84 HDAC3 (0.41) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL19545290 0.83 HDAC3 (0.40) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL19545291 0.75 MAPK1 (0.43) HDAC3HDAC1HDAC2NCOR2BACE1
SCHEMBL8329333 0.75 KDM1A (0.40) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL8330600 0.74 KDM1A (0.39) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL8328152 0.74 RIPK1 (0.38) ADRB2ADRB1ADRB3RIPK1NPC1
SCHEMBL4744310 0.74 SSTR4 (0.56) HDAC3HDAC1HDAC2NCOR2KCNQ4
SCHEMBL2897902 0.74 HDAC3 (0.46) HDAC3HDAC1HDAC2NCOR2KCNQ4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0760368-B1 PYRIMIDINE DERIVATIVES NISSHIN FLOUR MILLING CO (JP) 1999-07-28 EP disclosed
US-5736550-A TREATMENT OF GASTROINTESTINAL TRACT DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-04-07 US disclosed
EP-0760368-A1 NOVEL PYRIMIDINE DERIVATIVE NISSHIN FLOUR MILLING CO., LTD. (JP) 1997-03-05 EP disclosed