SCHEMBL8328694

SCHEMBL8328694

CS(=O)(=O)c1ccc(Nc2cncnc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PIP4K2C Q8TBX8 8/20 0.46
PIP4K2A P48426 5/20 0.46
TNNI3K Q59H18 1/20 0.43
GSK3B P49841 1/20 0.41
TGM2 P21980 1/20 0.41
ENPP2 Q13822 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25667539 0.84 ENPP2 (0.54) PIP4K2CPIP4K2AGSK3BTGM2ENPP2
SCHEMBL11882073 0.81 SOS1 (0.54)
SCHEMBL3245767 0.76 MEN1 (0.58) GSK3B
SCHEMBL2877698 0.75 GSK3B (0.59) GSK3B
SCHEMBL24383402 0.73 ENPP2 (0.43) PIP4K2CPIP4K2AGSK3BTGM2ENPP2
SCHEMBL5457984 0.73 ENPP2 (0.43) PIP4K2CPIP4K2ATNNI3KGSK3BTGM2
SCHEMBL4191619 0.73 XDH (0.54) PIP4K2AGSK3B
SCHEMBL28324029 0.73 TNNI3K (0.51) PIP4K2CPIP4K2ATNNI3K
SCHEMBL29501363 0.73 TNNI3K (0.51) PIP4K2CPIP4K2ATNNI3K
SCHEMBL12656068 0.73 ENPP2 (0.39) ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
CN-1039228-C Novel substituted tert-amino compund YAMANOUCHI PHARMA CO LTD (JP) 1998-07-22 CN disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed