SCHEMBL8328773

SCHEMBL8328773

Clc1ccc(-c2ncc3c(n2)-c2ncncc2CC3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.39
CYP1A2 P05177 3/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
CYP2C19 P33261 3/20 0.36
CYP2C9 P11712 2/20 0.36
CYP3A4 P08684 2/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP2D6 P10635 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
LMNA P02545 1/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329431 0.83 CCNA2 (0.44) HRH4CYP1A2USP2TSHRCYP2C19
SCHEMBL8326631 0.80 KDM4E (0.43) HRH4CYP1A2CYP2C19CYP2C9CYP3A4
SCHEMBL8329211 0.77 KDM4E (0.43) HRH4CYP1A2CYP2C19CYP2C9CYP3A4
SCHEMBL15750969 0.73 GABRG2 (0.33) RAB9AMAPTCDK2SMN1; SMN2
SCHEMBL8330251 0.72 DUSP10 (0.45) CYP1A2CYP2C19CYP2C9CYP3A4KDM4E
SCHEMBL8325184 0.71 CCNA2 (0.62) CYP1A2CYP2C19CYP2C9CYP3A4KDM4E
SCHEMBL8329082 0.71 CCNA2 (0.48) CYP1A2CYP2C19CYP2C9CYP3A4KDM4E
SCHEMBL8327052 0.70 CDK2 (0.35) CYP1A2CYP2C19CYP2C9CYP3A4KDM4E
SCHEMBL8327283 0.70 CYP2C19 (0.42) HRH4CYP1A2CYP2C19CYP2C9CYP3A4
SCHEMBL22966310 0.69 CYP19A1 (0.48) HRH4LMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP claimed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO claimed
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed