SCHEMBL8327052

SCHEMBL8327052

Clc1ccc(-c2ncc3c(n2)-c2cncnc2CC3)cn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.35
CCNA2 P20248 5/20 0.35
CCNT1 O60563 1/20 0.35
CDK1 P06493 1/20 0.35
CDK4 P11802 1/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK7 P50613 1/20 0.35
CDK9 P50750 1/20 0.35
CCNH P51946 1/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA4 P22748 1/20 0.34
CA9 Q16790 1/20 0.34
CYP2A6 P11509 1/20 0.33
PIK3CD O00329 1/20 0.32
CASP3 P42574 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329431 0.87 CCNA2 (0.44) CDK2CCNA2CA1CA2CA4
SCHEMBL8327878 0.85 CCNA2 (0.34) CDK2CCNA2CA1CA2CA4
SCHEMBL8326389 0.82 CCNT1 (0.39) CDK2CCNT1CDK1CDK4CCNB1
SCHEMBL8326151 0.81 CYP1A2 (0.41) CDK2CCNA2CYP2A6KDM4EALDH1A1
SCHEMBL8327742 0.74 CCNA2 (0.34) CDK2CCNA2CA1CA2CA4
SCHEMBL8325671 0.73 CCNA2 (0.40) CDK2CCNA2KDM4E
SCHEMBL8328773 0.70 HRH4 (0.39) CDK2CCNA2KDM4ECYP1A2CYP3A4
SCHEMBL8330251 0.69 DUSP10 (0.45) CDK2CCNA2KDM4EALDH1A1POLB
SCHEMBL8329211 0.69 KDM4E (0.43) CDK2CCNA2KDM4EALDH1A1POLB
SCHEMBL8329082 0.68 CCNA2 (0.48) CDK2CCNA2CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP claimed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO claimed
EP-0915879-A1 NOVEL COMPOUNDS Astra Pharmaceuticals Limited (GB) 1999-05-19 EP disclosed
WO-1998001449-A1 NOVEL COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1998-01-15 WO disclosed