SCHEMBL8328796

SCHEMBL8328796

CCOC(=O)C1=C(OC(C)=O)c2cc3ccccc3n2CC1C(=O)OCC

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOD2 Q9HC29 6/20 0.39
NOD1 Q9Y239 6/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
KDM4E B2RXH2 4/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
ADORA2B P29275 1/20 0.37
HPGD P15428 4/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CHRM1 P11229 1/20 0.35
CHRM3 P20309 1/20 0.35
ALDH1A1 P00352 2/20 0.35
F10 P00742 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KIF11 P52732 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326257 0.86 KDM4E (0.42) NOD2NOD1MEN1KMT2AKDM4E
SCHEMBL8655802 0.81 MAPT (0.44) NOD2NOD1MEN1KMT2AKDM4E
SCHEMBL8658440 0.75 KDM4E (0.40) NOD2NOD1MEN1KMT2AKDM4E
SCHEMBL8447552 0.68 ALDH1A1 (0.44) MEN1KMT2AKDM4ESMN1; SMN2ALDH1A1
SCHEMBL8328799 0.67 ATM (0.41) MEN1KMT2AKDM4ESMN1; SMN2HPGD
SCHEMBL18202192 0.67 HSD17B10 (0.38) KDM4EHPGDCHRM2CHRM4CHRM5
SCHEMBL8328343 0.66 ALDH1A1 (0.45) KDM4ESMN1; SMN2HPGDALDH1A1ATM
SCHEMBL8328857 0.66 SMN1; SMN2 (0.49) NOD2NOD1MEN1KMT2AKDM4E
SCHEMBL8657539 0.66 ALDH1A1 (0.47) MEN1KMT2AKDM4EHPGDALDH1A1
SCHEMBL9256630 0.66 MAPT (0.41) MEN1KMT2AKDM4ESMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed