SCHEMBL8328799

SCHEMBL8328799

CCOC(=O)C1=C(OC(C)=O)c2cc3ccccn3c2CC1C(=O)OCC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 2/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 8/20 0.38
KDM4E B2RXH2 4/20 0.38
HPGD P15428 3/20 0.38
GAA P10253 2/20 0.38
GLA P06280 1/20 0.38
MAPK1 P28482 3/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NPSR1 Q6W5P4 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 1/20 0.35
IDO1 P14902 1/20 0.35
HBB P68871 1/20 0.35
HIF1A Q16665 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8326264 0.86 ATM (0.43) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL8328861 0.70 L3MBTL1 (0.46) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL8328796 0.67 NOD2 (0.39) ATML3MBTL1ALDH1A1KDM4EHPGD
SCHEMBL17331983 0.67 L3MBTL1 (0.58) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL3150589 0.67 ATM (0.45) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL8328348 0.67 ATM (0.45) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL9430376 0.65 HTT (0.46) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL21239633 0.65 KDM4E (0.58) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL9430322 0.65 HTT (0.41) ATMHTTL3MBTL1ALDH1A1KDM4E
SCHEMBL9429930 0.64 HTT (0.44) ATMHTTL3MBTL1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470490-B1 Substituted pyrroles HOFFMANN LA ROCHE (CH) 1999-05-06 EP disclosed
US-5292747-A Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 1994-03-08 US disclosed
EP-0470490-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1992-02-12 EP disclosed