SCHEMBL8328937

SCHEMBL8328937

C=C(c1ccc([N+](=O)[O-])cc1)N(c1ccc(C#N)cc1)c1cncnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.42
THRB P10828 1/20 0.42
KCNJ1 P48048 1/20 0.37
KCNH2 Q12809 1/20 0.37
CYP19A1 P11511 3/20 0.36
PGR P06401 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
CARM1 Q86X55 1/20 0.34
PRMT1 Q99873 1/20 0.34
CES1 P23141 1/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
VCAM1 P19320 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8328528 0.80 MEN1 (0.49) MAPTTHRBKCNJ1KCNH2CYP19A1
SCHEMBL8324619 0.74 KCNJ1 (0.46) MAPTKCNJ1KCNH2CYP19A1PGR
SCHEMBL8323517 0.74 KCNJ1 (0.46) MAPTKCNJ1KCNH2CYP19A1PGR
SCHEMBL8330474 0.73 CYP19A1 (0.43) MAPTTHRBKCNJ1KCNH2CYP19A1
SCHEMBL31257790 0.70 MEN1 (0.61) MAPTTHRBKCNJ1KCNH2CYP19A1
SCHEMBL57257 0.70 VCAM1 (0.61) MAPTTHRBKCNJ1KCNH2PGR
SCHEMBL16089350 0.70 VCAM1 (0.61) MAPTTHRBKCNJ1KCNH2PGR
Selenium SCHEMBL9497333 0.68 VCAM1 (0.59) MAPTTHRBKCNJ1KCNH2PGR
SCHEMBL8327373 0.68 ALDH1A1 (0.61) MAPTCYP19A1L3MBTL1NPC1CES1
SCHEMBL6164603 0.68 MAPT (0.35) MAPTTHRBKCNJ1KCNH2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed
CN-1079962-A New substituted tertiary amine compound and salt thereof YAMANOUCHI PHARMA CO LTD (JP) 1993-12-29 CN disclosed