SCHEMBL8324619

SCHEMBL8324619

N#Cc1ccc(N(Cc2ccc([N+](=O)[O-])cc2)c2cncnc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 2/20 0.46
KCNH2 Q12809 2/20 0.46
NPC1 O15118 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.41
CYP19A1 P11511 2/20 0.40
AR P10275 9/20 0.39
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
PYCR1 P32322 1/20 0.39
POLB P06746 1/20 0.38
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
PGR P06401 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8323517 1.00 KCNJ1 (0.46) KCNJ1KCNH2NPC1MAPTPKM
SCHEMBL8327952 0.90 CRHBP (0.47) CYP19A1ARCRHBPCRHR2PYCR1
SCHEMBL8328066 0.87 CYP19A1 (0.44) CYP19A1ARCRHBPCRHR2POLB
SCHEMBL8323939 0.84 AR (0.49) KCNJ1KCNH2NPC1CYP19A1AR
SCHEMBL8327623 0.84 ALDH1A1 (0.50) NPC1MAPTCYP19A1ARCRHBP
SCHEMBL8326188 0.84 CYP19A1 (0.55) NPC1MAPTCYP19A1ARCRHBP
SCHEMBL8327171 0.84 CRHBP (0.42) MAPTCYP19A1ARCRHBPCRHR2
SCHEMBL8323116 0.82 CYP19A1 (0.39) MAPTCYP19A1POLB
SCHEMBL8328528 0.82 MEN1 (0.49) KCNJ1KCNH2NPC1MAPTPKM
SCHEMBL8329428 0.81 MAOA (0.42) CYP19A1CRHBPCRHR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640595-B1 SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMA CO LTD (JP) 1999-03-24 EP disclosed
US-5538976-A ANTICARCINOGENIC AGENTS AND ENZYME INHIBITORS FOR AROMATASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1996-07-23 US disclosed
EP-0640595-A1 NOVEL SUBSTITUTED TERTIARY AMINO COMPOUND OR SALT THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1995-03-01 EP disclosed