SCHEMBL8329202

SCHEMBL8329202

Cn1cccc1-c1cc(Cl)nc(N)n1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 9/20 0.55
HSP90AB1 P08238 9/20 0.55
KDM4E B2RXH2 1/20 0.51
ADCY10 Q96PN6 11/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29094518 0.83 ALOX15 (0.41) HSP90AA1HSP90AB1KDM4E
SCHEMBL29094466 0.77 ALOX15 (0.37) HSP90AA1HSP90AB1KDM4E
SCHEMBL29094580 0.76 ALOX15 (0.39) HSP90AA1HSP90AB1KDM4E
SCHEMBL3952089 0.70 HSP90AA1 (0.70) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL29571104 0.70 HSP90AA1 (0.70) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL22501986 0.69 HSP90AA1 (0.66) HSP90AA1HSP90AB1KDM4EADCY10
SCHEMBL439225 0.69 KDM4E (0.49) KDM4E
SCHEMBL29094509 0.69 ALDH1A1 (0.44) KDM4E
SCHEMBL1643108 0.68 HSP90AA1 (1.00) HSP90AA1HSP90AB1KDM4E
Hydrochloric Acid SCHEMBL22502036 0.68 HSP90AA1 (0.64) HSP90AA1HSP90AB1KDM4EADCY10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7737153-B2 Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-15 US disclosed
US-7737153-B2 Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-06-15 US disclosed
WO-2004039796-A1 HETEROARYLOXY-SUBSTITUTED PHENYLAMINOPYRIMIDINES AS RHO-KINASE INHIBITORS BAYER HEALTHCARE AG (DE) 2004-05-13 WO disclosed