SCHEMBL8329361

SCHEMBL8329361

CCc1cccc(C(C)C(=O)N(C)C2CC2)c1

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 7/20 0.49
PTGS2 P35354 1/20 0.44
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALOX5 P09917 1/20 0.39
DPP4 P27487 1/20 0.39
DPP9 Q86TI2 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SMYD3 Q9H7B4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331069 0.86 CCR5 (0.39) CCR5PTGS2SMN1; SMN2DPP4DPP9
SCHEMBL4682033 0.77 PTGS2 (0.51) PTGS2AKR1C3AKR1C2SMN1; SMN2ALOX5
SCHEMBL3674499 0.76 PTGS2 (0.69) PTGS2AKR1C3AKR1C2SMN1; SMN2ALOX5
SCHEMBL1691998 0.75 SMYD3 (0.49) CCR5SMN1; SMN2MEN1KMT2ASMYD3
SCHEMBL8335577 0.75 SMYD3 (0.52) PTGS2SMN1; SMN2SMYD3
SCHEMBL4682035 0.74 PTGS2 (0.51) PTGS2AKR1C3AKR1C2SMN1; SMN2
SCHEMBL8333192 0.71 KCNQ2 (0.46) CCR5DPP4DPP9MEN1KMT2A
SCHEMBL6036650 0.71 PTGS2 (0.41) PTGS2AKR1C3AKR1C2SMN1; SMN2MEN1
SCHEMBL17896334 0.70 CCR5 (0.55) CCR5KMT2A
SCHEMBL8332307 0.70 ACHE (0.43) CCR5DPP4DPP9MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed