SCHEMBL8329530

SCHEMBL8329530

CCOC(=O)c1ccc(CCc2cc3c(cc2F)SC(C)(C)CC3=O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.39
PTPN1 P18031 1/20 0.38
MAPT P10636 6/20 0.38
MEN1 O00255 4/20 0.38
HPGD P15428 3/20 0.38
KDM4E B2RXH2 3/20 0.38
HIF1A Q16665 2/20 0.38
MAPK1 P28482 1/20 0.38
KCNJ1 P48048 1/20 0.37
KCNH2 Q12809 1/20 0.37
POLB P06746 1/20 0.36
CCR6 P51684 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
ALDH1A1 P00352 3/20 0.36
TSHR P16473 1/20 0.36
DRD2 P14416 1/20 0.36
DRD3 P35462 1/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8329526 0.80 MAPK1 (0.37) KMT2AMAPTMEN1HPGDKDM4E
SCHEMBL6589030 0.80 PRKCA (0.39) KMT2APTPN1MAPTMEN1HPGD
SCHEMBL727818 0.74 CYP3A4 (0.46) KMT2AMAPTMEN1HPGDKDM4E
SCHEMBL6591370 0.72 KMT2A (0.41) KMT2APTPN1MAPTMEN1HPGD
SCHEMBL8329533 0.70 ALDH1A1 (0.45) KMT2APTPN1MAPTMEN1HPGD
SCHEMBL16687963 0.70 CA12 (0.58) KMT2APTPN1MAPTMEN1HPGD
SCHEMBL6591091 0.70 KMT2A (0.38) KMT2AMEN1KDM4EALDH1A1RARA
SCHEMBL12199135 0.69 CA1 (0.68) KMT2APTPN1MAPTMEN1HPGD
SCHEMBL10765170 0.66 CYP4A11 (0.62) MAPTHPGDKDM4EHIF1AMAPK1
SCHEMBL16687614 0.65 CA2 (0.50) KMT2APTPN1MAPTMEN1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958954-A 2,2-DIALKYL-4-ARYL-SUBSTITUTED BENZOPYRAN AND BENZOTHIOPYRAN DERIVATIVES ALLERGAN SALES, INC. (US) 1999-09-28 US disclosed