SCHEMBL8329614

SCHEMBL8329614

Cc1nc2n(CC(O)c3ccccc3)cc(Cl)cc-2c1CC#N

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.36
PKM P14618 2/20 0.35
IDO1 P14902 1/20 0.34
TSHR P16473 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.32
GAA P10253 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
KDM4E B2RXH2 1/20 0.31
RET P07949 2/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
DPP4 P27487 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8327462 0.76 TSHR (0.39) ALDH1A1PKMIDO1TSHRGAA
SCHEMBL8326439 0.71 ALDH1A1 (0.42) ALDH1A1PKMIDO1TSHRGAA
Bromide SCHEMBL8327518 0.65 MEN1 (0.38) ALDH1A1GAALMNAHTT
SCHEMBL4259200 0.63 PRMT5 (0.57) ALDH1A1PKMTSHRSMN1; SMN2LMNA
SCHEMBL8325690 0.63 ATP4A (0.47) GAAKDM4EHTT
SCHEMBL8329254 0.63 CYP11B1 (0.35) ALDH1A1PKMTSHRGAAKDM4E
SCHEMBL8329568 0.58 KDM4E (0.39) PKMIDO1TSHRKDM4EHTT
SCHEMBL9130426 0.58 IDO1 (0.47) ALDH1A1PKMIDO1TSHRGAA
SCHEMBL11518221 0.58 ALDH1A1 (0.52) ALDH1A1PKMTSHRGAASMN1; SMN2
SCHEMBL31292178 0.56 DPP4 (0.32) ALDH1A1KDM4ELMNAHTTDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509974-B1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof ASTRA AB (SE) 1999-01-13 EP disclosed
US-5439917-A Phenyl-pyrrolo(2,3-b)pyridine antisecretory agent of gastric acid; adenosine triphosphatase enzyme inhibitor AKTIEBOLAGET ASTRA (SE) 1995-08-08 US disclosed
EP-0580616-A1 NEW ACTIVE COMPOUNDS Astra Aktiebolag (SE) 1994-02-02 EP disclosed
EP-0509974-A1 Pyrrolo[2,3-b]pyridines having therapeutic activity and a process for the preparation thereof Astra Aktiebolag (SE) 1992-10-21 EP disclosed
WO-1992017477-A1 NEW ACTIVE COMPOUNDS AKTIEBOLAGET ASTRA (SE) 1992-10-15 WO disclosed