SCHEMBL8329624

SCHEMBL8329624

O=[N+]([O-])c1ccc(CN2CCCCCCCCNNN2)cc1

nearest known ligand 0.57

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.46
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 4/20 0.44
MAPT P10636 3/20 0.44
LMNA P02545 2/20 0.44
KCNJ1 P48048 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNH2 Q12809 2/20 0.43
DBH P09172 1/20 0.42
CASP1 P29466 1/20 0.41
CASP4 P49662 1/20 0.41
CASP5 P51878 1/20 0.41
GBA1 P04062 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8790806 0.79 SIGMAR1 (0.42) HRH3ALDH1A1MAPTLMNA
SCHEMBL8790515 0.75 SIGMAR1 (0.41) HRH3ALDH1A1MAPTLMNA
SCHEMBL1805498 0.74 KDM4E (0.71) HRH3KDM4EALDH1A1MAPTLMNA
SCHEMBL3143167 0.74 KDM4E (0.71) HRH3KDM4EALDH1A1MAPTLMNA
SCHEMBL8329627 0.74 KDM4E (0.71) HRH3KDM4EALDH1A1MAPTLMNA
SCHEMBL2206628 0.72 KDM4E (0.73) HRH3KDM4EALDH1A1MAPTLMNA
SCHEMBL28801541 0.71 ALDH1A1 (0.50) KDM4EALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL27171599 0.71 KCNJ1 (0.58) HRH3KDM4EALDH1A1MAPTLMNA
SCHEMBL1022743 0.69 SIGMAR1 (0.44) HRH3ALDH1A1MAPTLMNA
SCHEMBL3156886 0.69 KDM4E (0.73) HRH3KDM4EALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0736035-A4 PRETARGETING METHODS AND COMPOUNDS NEORX CORP (US) 1999-09-01 EP disclosed
US-5847121-A Production of nitro-benzyl-dota via direct peptide cyclization NEORX CORPORATION (US) 1998-12-08 US disclosed
EP-0736035-A1 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1996-10-09 EP disclosed
US-5541287-A DIAGNOSIS USING CYCLIC TRIPEPTIDES WITH NITROBENZYL 1,4,7,10-TETRAAZACYCLODODECANE-N,N*,N**,N***TETRAACETIC ACID BIOTIN CONJUGATE FORMED BY ALKYLATION AND MULTISTAGE PROCESS NEORX CORPORATION (US) 1996-07-30 US disclosed
WO-1995015335-A2 PRETARGETING METHODS AND COMPOUNDS NEORX CORPORATION (US) 1995-06-08 WO disclosed