SCHEMBL8330002

SCHEMBL8330002

CCn1c(C(=O)O)cc(=O)cc1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 2/20 0.53
POLB P06746 5/20 0.40
KDM4E B2RXH2 5/20 0.40
PKM P14618 1/20 0.40
SRC P12931 1/20 0.39
ALDH1A1 P00352 6/20 0.37
HPGD P15428 4/20 0.37
HSD17B10 Q99714 3/20 0.37
TSHR P16473 2/20 0.37
BLM P54132 2/20 0.37
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
HASPIN Q8TF76 1/20 0.37
ALOX15 P16050 1/20 0.37
NFKB1 P19838 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CCR2 P41597 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.35
FDPS P14324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4957913 0.75 GPR35 (0.50) GPR35POLBKDM4EPKMALDH1A1
SCHEMBL11559372 0.75 POLB (0.43) POLBKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL1919417 0.72 GPR35 (0.47) GPR35KDM4ECCR2KMT2A
SCHEMBL10693316 0.72 POLB (0.37) GPR35POLBKDM4EPKMALDH1A1
SCHEMBL30067600 0.70 CCR2 (0.69) GPR35POLBALDH1A1TSHRCCR2
SCHEMBL701976 0.70 CCR2 (0.69) GPR35POLBALDH1A1TSHRCCR2
SCHEMBL14702784 0.70 GPR35 (1.00) GPR35POLBKDM4EPKMSRC
SCHEMBL17477638 0.69 GPR35 (0.41) GPR35POLBKDM4EPKMALDH1A1
SCHEMBL31094809 0.69 GPR35 (0.45) GPR35POLBKDM4EPKMSRC
SCHEMBL1006638 0.69 GPR35 (0.44) GPR35POLBKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972975-A Substituted 2-aminopyridines as inhibitors of nitric oxide synthase MERCK & CO., INC. (US) 1999-10-26 US disclosed
WO-1996018616-A1 SUBSTITUTED 2-AMINOPYRIDINES AS INHIBITORS OF NITRIC OXIDE SYNTHASE MERCK & CO., INC. (US) 1996-06-20 WO disclosed