SCHEMBL8332822

SCHEMBL8332822

CC(CCC(N)=O)C1CC1c1cccc(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.46
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
ALOX5 P09917 2/20 0.41
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
HRH3 Q9Y5N1 1/20 0.37
RCOR1 Q9UKL0 1/20 0.36
TSHR P16473 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PARP1 P09874 1/20 0.35
HDAC4 P56524 1/20 0.34
F2RL1 P55085 1/20 0.33
DRD2 P14416 1/20 0.33
DRD1 P21728 1/20 0.33
DRD4 P21917 1/20 0.33
DRD5 P21918 1/20 0.33
DRD3 P35462 1/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331076 0.88 KDM1A (0.49) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8331361 0.86 HTR2A (0.45) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8331608 0.86 HTR2A (0.45) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8332794 0.85 SLC9A1 (0.47) HTR2AHTR2CHTR2BALOX5
SCHEMBL8331485 0.85 HTR2A (0.44) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8329354 0.83 SLC9A1 (0.51) HTR2AHTR2CHTR2BALOX5TSHR
SCHEMBL8334103 0.81 KDM1A (0.48) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8330436 0.80 KDM1A (0.51) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8716294 0.76 ALOX5 (0.34) KDM1AHTR2AHTR2CHTR2BALOX5
SCHEMBL8716974 0.74 SLC6A2 (0.36) KDM1AALOX5SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed