SCHEMBL8330462

SCHEMBL8330462

O=C1Nc2c(ccc3c2CN(Cc2ccccc2)C3)/C1=N/O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.38
TSHR P16473 1/20 0.38
KMT2A Q03164 1/20 0.38
ACHE P22303 2/20 0.36
PNMT P11086 1/20 0.36
KCNH2 Q12809 1/20 0.35
HDAC1 Q13547 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 1/20 0.35
SIGMAR1 Q99720 3/20 0.34
CYP1A2 P05177 1/20 0.34
PTGS2 P35354 1/20 0.34
BCHE P06276 1/20 0.34
IKZF2 Q9UKS7 1/20 0.34
DRD2 P14416 1/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8330468 1.00 MEN1 (0.38) MEN1TSHRKMT2AACHEPNMT
SCHEMBL8330647 0.84 BCHE (0.43) KMT2AACHEPNMTKDM4EALDH1A1
SCHEMBL8331247 0.83 PNMT (0.30) PNMT
SCHEMBL8331250 0.83 PNMT (0.30) PNMT
SCHEMBL8328966 0.76 ALDH1A1 (0.30) ALDH1A1
SCHEMBL3841662 0.76 SLC6A5 (0.42) MEN1KMT2AHDAC1DRD2SLC6A5
SCHEMBL8328965 0.76 ALDH1A1 (0.30) ALDH1A1
SCHEMBL3838812 0.76 SLC6A5 (0.42) MEN1KMT2AHDAC1DRD2SLC6A5
SCHEMBL8330987 0.73
SCHEMBL8329016 0.73 ALDH1A1 (0.31) ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529636-B1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH AS (DK) 1999-06-23 EP disclosed
US-5436250-A Isatineoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1995-07-25 US disclosed
US-5242918-A Isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-09-07 US disclosed
WO-1993005043-A1 NOVEL ISATINOXIME DERIVATIVES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 1993-03-18 WO disclosed
EP-0529636-A1 Novel isatinoxime derivatives, their preparation and use NEUROSEARCH A/S (DK) 1993-03-03 EP disclosed