SCHEMBL8334103

SCHEMBL8334103

CC(CCC(N)=O)C1CC1c1ccc(Br)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 11/20 0.48
KCNH2 Q12809 2/20 0.48
KDM1B Q8NB78 2/20 0.48
SLC9A1 P19634 1/20 0.39
RCOR1 Q9UKL0 1/20 0.38
ALOX5 P09917 2/20 0.34
KIF11 P52732 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716294 0.86 ALOX5 (0.34) KDM1ASLC9A1ALOX5HTR2AHTR2C
SCHEMBL8333860 0.81 KDM1A (0.35) KDM1AKCNH2KDM1BHTR2AHTR2C
SCHEMBL8332822 0.81 KDM1A (0.46) KDM1ARCOR1ALOX5HTR2AHTR2C
SCHEMBL8331485 0.81 HTR2A (0.44) KDM1ARCOR1ALOX5HTR2AHTR2C
SCHEMBL8335022 0.77 KDM1A (0.47) KDM1AKDM1BHTR2AHTR2CHTR2B
SCHEMBL8331608 0.77 HTR2A (0.45) KDM1AALOX5HTR2AHTR2CHTR2B
SCHEMBL8331361 0.77 HTR2A (0.45) KDM1AALOX5KIF11HTR2AHTR2C
SCHEMBL8332794 0.76 SLC9A1 (0.47) SLC9A1ALOX5HTR2AHTR2CHTR2B
SCHEMBL8716974 0.74 SLC6A2 (0.36) KDM1AALOX5
SCHEMBL8332303 0.74 ADAM17 (0.38) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5889031-A CONTROLLING CIRCADIAN RHYTHMS BRISTOL-MYERS SQUIBB COMPNAY (US) 1999-03-30 US disclosed
US-5753709-A N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics BRISTOL-MYERS SQUIBB COMPANY (US) 1998-05-19 US disclosed