SCHEMBL8334

SCHEMBL8334

O=C(O)N1CCC(n2cc(Br)c(=O)[nH]c2=O)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
POLB P06746 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TK1 P04183 1/20 0.39
PYGM P11217 1/20 0.39
GRIA1 P42261 1/20 0.37
GRIA2 P42262 1/20 0.37
GRIA4 P48058 1/20 0.37
GRIK5 Q16478 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PNP P00491 1/20 0.35
CALCRL Q16602 2/20 0.34
TNKS O95271 1/20 0.34
GAA P10253 1/20 0.34
SQOR Q9Y6N5 1/20 0.33
DRD2 P14416 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
RAMP1 O60894 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14193 0.82 SRC (0.44) ALDH1A1POLBKMT2ASMN1; SMN2
SCHEMBL28630594 0.75 SLC28A1 (0.37) PNPCALCRLRAMP1
SCHEMBL28630591 0.75 SLC28A1 (0.37) PNPCALCRLRAMP1
SCHEMBL12062409 0.75 ALDH1A1 (0.60) ALDH1A1POLBKMT2ASMN1; SMN2TK1
SCHEMBL19513999 0.72 KDM5A (0.42) ALDH1A1POLBKMT2ASMN1; SMN2GAA
SCHEMBL28539787 0.72 KDM5A (0.42) ALDH1A1POLBKMT2ASMN1; SMN2GAA
SCHEMBL3250125 0.69 DRD2 (0.37) KMT2ACALCRLTNKSDRD2DRD4
SCHEMBL3246969 0.69 CALCRL (0.45) CALCRLTNKSDRD2DRD4DRD3
SCHEMBL2099353 0.68 DRD2 (0.65) CALCRLTNKSDRD2DRD4DRD3
SCHEMBL28541089 0.67 KDM5A (0.54) ALDH1A1KMT2ASMN1; SMN2TDP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488525-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME Rib-X Pharmaceuticals, Inc. (US) 2012-08-22 EP disclosed
WO-2011047319-A2 ANTIMICROBIAL COMPOUNDS AND METHODS OF MAKING AND USING THE SAME RIB-X PHARMACEUTICALS, INC. (US) 2011-04-21 WO disclosed