SCHEMBL8334072

SCHEMBL8334072

CC(C)(c1ccccc1)c1cc(-c2cccc3nn(O)nc23)cc(C(C)(C)c2ccccc2)c1

nearest known ligand 0.37

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.37
CNR2 P34972 4/20 0.37
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28511468 0.92 CNR1 (0.45) CNR1CNR2ESR1ESR2ALDH1A1
SCHEMBL28608544 0.82 KIF11 (0.43)
SCHEMBL28461145 0.82 NPC1 (0.35)
SCHEMBL1263567 0.78 MET (0.38) ALDH1A1
SCHEMBL5474544 0.74 CNR1 (0.37) CNR1CNR2ESR1ESR2ALDH1A1
SCHEMBL1643503 0.72 ENPP1 (0.41) ALDH1A1
SCHEMBL8855679 0.71 CNR1 (0.38) CNR1CNR2ESR1ESR2ALDH1A1
SCHEMBL8645604 0.71 COMT (0.39) ALDH1A1
SCHEMBL8680274 0.71 CNR1 (0.40) CNR1CNR2ESR1ESR2ALDH1A1
SCHEMBL6445924 0.69 KDM4E (0.52) CNR1CNR2ESR1ESR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5952096-A CONSISTS OF POLYCARBONATE RESIN, TWO ULTRAVIOLET ABSORBERS OF SPECIFIC ABSORPTION WAVELENGTHS; EXCELLENT IMPACT STRENGTH, TRANSPARENCY AND HIGH ABSORPTION POWER FOR ULTRAVIOLET LIGHT HAVING A SPECIFIC WAVELENGTH TEIJIN CHEMICALS, LTD. (JP) 1999-09-14 US claimed
US-5852087-A Easily dyeable meta-linkage-containing aromatic polyamide fibers TEIJIN LIMITED (JP) 1998-12-22 US claimed
US-5849821-A Tris-aryl-s-triazines substituted with biphenylyl groups CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-12-15 US claimed
US-5958637-A CHARGE GENERATING LAYER CONTAINING PHTHALOCYANINE COMPOSITION AND CHARGE TRANSPORT MATERIAL COMPRISING A BENZIDINE DERIVATIVE HITACHI CHEMICAL COMPANY, LTD. (JP) 1999-09-28 US disclosed
US-5952096-A CONSISTS OF POLYCARBONATE RESIN, TWO ULTRAVIOLET ABSORBERS OF SPECIFIC ABSORPTION WAVELENGTHS; EXCELLENT IMPACT STRENGTH, TRANSPARENCY AND HIGH ABSORPTION POWER FOR ULTRAVIOLET LIGHT HAVING A SPECIFIC WAVELENGTH TEIJIN CHEMICALS, LTD. (JP) 1999-09-14 US disclosed
US-5948844-A ALIPHATIC CARBOXYLIC ACID METAL SALT IS ADDED TO A TERMINALLY STABILIZED POLYACETAL RESIN, SAID SALT HAVING OCCLUDED THEREIN AT LEAST ONE METAL COMPOUND SELECTED FROM THE GROUP CONSISTING OF A METAL HYDROXIDE AND A METAL CHLORIDE ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1999-09-07 US disclosed
US-5942626-A REACTING A 5-HALO-SUBSTITUTED BENZOTRIAZOLE WITH A MERCAPTO COMPOUND IN THE PRESENCE OF A GROUP 1A METAL OR GROUP 2A COMPOUND FORMING 5-THIO-SUBSTITUTED 2H-BENZOTRIAZOLES HAVING ENHANCED ABSORBANCE AT LONGER WAVELENGTHS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-08-24 US disclosed
US-5922794-A SYNERGISTIC COMBINATION OF TERTIARY AMINE OXIDE AND OTHER STABILIZERS TO PROVIDE DISCOLORATION AND HEAT RESISTANCE TO THERMOPLASTIC RESINS GENERAL ELECTRIC COMPANY (US) 1999-07-13 US disclosed
US-5891235-A RESIN PLUS ALUMINUM SILICATES MIZUSAWA INDUSTRIAL CHEMICALS, LTD. (JP) 1999-04-06 US disclosed
US-5889100-A POLYMER BLEND; MOLDING MATERIAL JAPAN POLYOLEFINS CO., LTD. (JP) 1999-03-30 US disclosed
US-5852087-A Easily dyeable meta-linkage-containing aromatic polyamide fibers TEIJIN LIMITED (JP) 1998-12-22 US disclosed
US-5807914-A POLYCARBONATE OLIGOMER, POLYSILOXANE-POLYACRYLATE COMPOSITE RUBBER GRAFTED WITH ACRYLONITRILE AND STYRENE MITSUBISHI ENGINEERING-PLASTICS CORPORATION (JP) 1998-09-15 US disclosed
US-5744527-A SHELL, CORE POLYMER POLYPLASTICS CO., LTD. (JP) 1998-04-28 US disclosed
US-5726309-A ULTRAVIOLET RADIATION ABSORBERS; THERMAL STABILIZERS FOR POLYMER SUBSTRATES, ESPECIALLY AUTOMOTIVE COATINGS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-03-10 US disclosed
US-5688592-A Thermochromic laminate comprising light intercepting pigment and light stabilizer THE PILOT INK CO., LTD. (JP) 1997-11-18 US disclosed
US-5684070-A FILM WITH TRIAZINE RESORCINOL COMPOUND STABILIZERS FOR RADIATION RESISTANCE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1997-11-04 US disclosed
US-5681955-A PHOTOSTABILITY OF POLYMERS CIBA SPECIALTY CHEMICALS CORPORATION (US) 1997-10-28 US disclosed
US-5679794-A ACTINIC LIGHT RESISTANCE, PROCESSING HEAT RESISTANCE CIBA-GEIGY CORPORATION (US) 1997-10-21 US disclosed
US-5674952-A FORMING POLYAMIDE, FORMING MELT POLYMER, APPLYING SHEAR, FORMING PARISON, BLOW MOLDING TORAY INDUSTRIES, INC. (JP) 1997-10-07 US disclosed
US-5675004-A POLYMER STABILIZERS TO PROTECT AGAINST ACTINIC RADIATION COVERING MORE OF THE NEAR-UV SPECTRUM; DISCOLORATION INHIBITION; SYNERGISTIC EFFECT WITH HINDERED AMINES; ALKYD, ACRYLIC, URETHANE COATINGS CIBA-GEIGY CORPORATION (US) 1997-10-07 US disclosed