SCHEMBL8335648

SCHEMBL8335648

CN(C)c1cccc(NC(=O)C(NC(=O)OC(C)(C)C)c2ccccc2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.54
CTSK P43235 1/20 0.54
BACE1 P56817 4/20 0.52
HDAC4 P56524 2/20 0.47
HDAC1 Q13547 2/20 0.47
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
KDM4E B2RXH2 3/20 0.46
TDP1 Q9NUW8 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31048635 0.86 CTSK (0.66) CTSSCTSKBACE1HDAC4HDAC1
SCHEMBL8338149 0.86 CTSK (0.66) CTSSCTSKBACE1HDAC4HDAC1
SCHEMBL8336972 0.85 CTSS (0.57) CTSSCTSKBACE1HDAC4HDAC1
SCHEMBL6726960 0.85 ALDH1A1 (0.51) BCHEACHEKDM4ETDP1ALDH1A1
SCHEMBL8337364 0.82 SMN1; SMN2 (0.58) CTSSCTSKBACE1KDM4EHDAC8
SCHEMBL8336482 0.82 SMN1; SMN2 (0.58) CTSSCTSKBACE1KDM4EHDAC8
SCHEMBL6715868 0.81 CTSS (0.57) CTSSCTSKBACE1KDM4EHDAC8
SCHEMBL8338577 0.81 CTSS (0.57) CTSSCTSKBACE1HDAC4HDAC1
SCHEMBL8337969 0.81 CTSS (0.57) CTSSCTSKBACE1HDAC4HDAC1
SCHEMBL16709839 0.80 BCHE (0.56) HDAC1BCHEACHEHDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022528-A2 ARYLGLYCINE DERIVATIVES AND THEIR USE AS GLYCINE TRANSPORT INHIBITORS NPS ALLELIX CORP. (CA) 2004-03-18 WO disclosed