SCHEMBL8338716

SCHEMBL8338716

COc1cccc(-c2cc(OCCBr)cc(C)c2C(=O)c2csc3ccccc23)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.40
HTR1D P28221 1/20 0.37
CNR2 P34972 2/20 0.37
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8339556 0.92 MAPT (0.38) HTR1AHTR1DCNR2MAPTKDM4E
SCHEMBL8339230 0.91 TUBB4A (0.40) HTR1AHTR1DCNR2MAPTKDM4E
SCHEMBL8334595 0.91 CNR2 (0.39) HTR1ACNR2MAPTMEN1CYP1A2
SCHEMBL8335086 0.88 CNR2 (0.36) HTR1ACNR2MAPTCYP1A2CYP2C19
SCHEMBL8340536 0.87 CNR2 (0.36) HTR1ACNR2MAPTMEN1CYP1A2
SCHEMBL8339826 0.86 KDM4E (0.42) HTR1AHTR1DCNR2MAPTKDM4E
SCHEMBL8340220 0.86 PRKCZ (0.41) HTR1AHTR1DMAPTKDM4EMEN1
SCHEMBL8341645 0.85 TUBB4A (0.40) HTR1AHTR1DCNR2MAPTKDM4E
SCHEMBL8339938 0.85 PRKCZ (0.40) HTR1ACNR2MAPTKDM4EMEN1
SCHEMBL8336646 0.85 CNR2 (0.35) HTR1ACNR2MAPTCYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948796-A OSTEOPOROSIS, CANCER, CARDIOVASCULAR DISORDERS ELI LILLY AND COMPANY (US) 1999-09-07 US disclosed