SCHEMBL8339265

SCHEMBL8339265

[c]1ccccc1CNOCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRAS P01112 1/20 0.47
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
TSHR P16473 2/20 0.38
IDO1 P14902 3/20 0.35
BCHE P06276 3/20 0.35
AGXT P21549 1/20 0.34
THRB P10828 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206646 0.77 HRAS (0.65) HRASNPC1RAB9ATSHRIDO1
SCHEMBL10776729 0.75 HRAS (0.68) HRASNPC1RAB9ATSHRIDO1
Hydrochloric Acid SCHEMBL6967279 0.75 HRAS (0.62) HRASNPC1RAB9ATSHRIDO1
SCHEMBL8339266 0.75 HRAS (0.54) HRASNPC1RAB9ATSHRIDO1
SCHEMBL6999395 0.74 TSHR (0.60) TSHRIDO1AGXT
SCHEMBL2650327 0.74 MEN1 (0.50) IDO1BCHETHRBMEN1KMT2A
SCHEMBL11116669 0.73 LMNA (0.54) NPC1RAB9A
SCHEMBL8340179 0.71 TSHR (0.40) HRASNPC1RAB9ATSHRIDO1
SCHEMBL6330694 0.70 ALDH1A1 (0.43) MEN1KMT2A
SCHEMBL8333710 0.69 TSHR (0.38) NPC1RAB9ATSHRIDO1AGXT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877312-A Method for preparing alkylating agents for their use for alkylating cyclic ureas DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-02 US claimed
US-5637780-A Method for preparing alkylating agents and their use for alkylating cyclic ureas THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-06-10 US claimed
EP-0767770-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-04-16 EP claimed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO claimed
US-5877312-A Method for preparing alkylating agents for their use for alkylating cyclic ureas DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-02 US disclosed
US-5637780-A Method for preparing alkylating agents and their use for alkylating cyclic ureas THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-06-10 US disclosed
EP-0767770-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-04-16 EP disclosed
WO-1996000708-A1 METHOD FOR PREPARING ALKYLATING AGENTS AND THEIR USE FOR ALKYLATING CYCLIC UREAS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-11 WO disclosed