SCHEMBL8339658

SCHEMBL8339658

O=C(NCc1ccccc1O)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.70
HTT P42858 1/20 0.65
EPHX2 P34913 3/20 0.60
NR1H4 Q96RI1 1/20 0.60
EGFR P00533 2/20 0.59
HDAC3 O15379 1/20 0.59
HDAC4 P56524 1/20 0.59
HDAC1 Q13547 1/20 0.59
HDAC7 Q8WUI4 1/20 0.59
HDAC2 Q92769 1/20 0.59
HDAC10 Q969S8 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
HDAC9 Q9UKV0 1/20 0.59
HDAC5 Q9UQL6 1/20 0.59
MMP13 P45452 1/20 0.57
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
HIF1A Q16665 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30646449 0.90 HPGD (0.67) SMN1; SMN2HTTHDAC1HDAC6HIF1A
SCHEMBL5723909 0.90 HPGD (0.67) SMN1; SMN2HTTHDAC1HDAC6HIF1A
SCHEMBL14817912 0.84 ALDH1A1 (0.51) SMN1; SMN2HTTHDAC1HIF1ACA2
SCHEMBL12459658 0.84 CA2 (0.52) SMN1; SMN2HTTEPHX2NR1H4HDAC1
SCHEMBL14817978 0.84 ALDH1A1 (0.59) SMN1; SMN2HTTHDAC3HDAC1NPC1
SCHEMBL539059 0.80 EPHX2 (0.84) SMN1; SMN2EPHX2NR1H4EGFRHDAC3
SCHEMBL4926867 0.77 CYP2D6 (0.50) SMN1; SMN2NPC1HIF1ACA2ALDH1A1
SCHEMBL4839587 0.77 TSHR (0.59) HTTHIF1ACA2ALDH1A1HPGD
SCHEMBL3389986 0.76 HPGD (0.57) SMN1; SMN2HTTNPC1HIF1ALMNA
SCHEMBL21812516 0.75 EGFR (0.57) SMN1; SMN2HTTEPHX2NR1H4EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014844-A2 ARYL AND HETEROARYL COMPOUNDS AND METHODS TO MODULATE COAGULATION TRANSTECH PHARMA, INC. (US) 2004-02-19 WO disclosed