SCHEMBL8340646

SCHEMBL8340646

Cn1c(=O)n(Cc2ccc(F)c(F)c2)c(=O)c2cc(C(=O)O)[nH]c21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.41
PTGS2 P35354 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.40
GPR18 Q14330 1/20 0.40
LGMN Q99538 1/20 0.39
PDE3B Q13370 5/20 0.38
PDE3A Q14432 5/20 0.38
MMP13 P45452 1/20 0.38
SLC22A8 Q8TCC7 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
GRIN1 Q05586 2/20 0.36
GRIN2B Q13224 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6684759 0.86 ALDH1A1 (0.41) PTGS1PTGS2PTGDR2GPR18PDE3B
SCHEMBL6682303 0.85 S1PR3 (0.47) GPR18
SCHEMBL8340699 0.83 PDE3B (0.43) PTGS1PTGS2GPR18LGMNPDE3B
SCHEMBL6703216 0.78 ADORA2B (0.38) PTGS1PTGS2PTGDR2GPR18LGMN
SCHEMBL6843728 0.77 MMP13 (0.48) PTGS1PTGS2GPR18LGMNPDE3B
SCHEMBL6466057 0.76 MMP13 (0.57) PTGS1PTGS2PTGDR2MMP13SLC22A8
SCHEMBL6698891 0.76 PTGS1 (0.41) PTGS1PTGS2PTGDR2GPR18MMP13
SCHEMBL6703224 0.76 PTGS1 (0.41) PTGS1PTGS2PTGDR2GPR18MMP13
SCHEMBL7018972 0.74 GRIN1 (0.44) PTGS1PTGS2PTGDR2MMP13SLC22A8
SCHEMBL6735485 0.72 LGMN (0.48) LGMNPDE3BPDE3AMMP13SLC22A8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004014384-A2 CYCLIC COMPOUNDS CONTAINING ZINC BINDING GROUPS AS MATRIX METALLOPROTEINASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2004-02-19 WO disclosed