SCHEMBL8340938

SCHEMBL8340938

CC(C)(C)Cc1ccc(N2C=NCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.40
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
SLC6A2 P23975 1/20 0.31
HTR2A P28223 1/20 0.31
SLC6A4 P31645 1/20 0.31
HRH1 P35367 1/20 0.31
HTR2B P41595 1/20 0.31
CHRNA4 P43681 1/20 0.31
SLC6A3 Q01959 1/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14536064 0.81 NPC1 (0.41) THRB
SCHEMBL28259847 0.70 KIF11 (0.39)
SCHEMBL6272216 0.70 SIGMAR1 (0.41) CHRNA4
SCHEMBL105023 0.70 SIGMAR1 (0.41) CHRNA4
SCHEMBL28131603 0.70 CHKA (0.46)
SCHEMBL11923149 0.69 ALDH1A1 (0.48) ESR1THRB
SCHEMBL28261625 0.69 LMNA (0.45) HRH1
SCHEMBL6685103 0.68 ESR1 (0.74) ESR1THRATHRBSLC6A2HTR2A
SCHEMBL13007692 0.68 ALDH1A1 (0.52) ESR1THRB
SCHEMBL7729842 0.67 MAPT (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004043367-A2 FUSED HETEROCYCLIC COMPOUNDS AND USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2004-05-27 WO disclosed