SCHEMBL8345834

SCHEMBL8345834

COC(=O)CCC(c1cnc2c(c1)CCCC2)C1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
GPR119 Q8TDV5 10/20 0.40
DPP4 P27487 1/20 0.38
MMP13 P45452 5/20 0.37
EED O75530 1/20 0.37
RBBP4 Q09028 1/20 0.37
SUZ12 Q15022 1/20 0.37
EZH2 Q15910 1/20 0.37
AEBP2 Q6ZN18 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
MMP1 P03956 3/20 0.36
MMP3 P08254 3/20 0.36
MMP7 P09237 3/20 0.36
MMP9 P14780 3/20 0.36
MMP8 P22894 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12892140 0.91 NPC1 (0.41) NPC1RAB9AGPR119DPP4MMP13
SCHEMBL8345088 0.81 ITGB3 (0.48) NPC1RAB9AGPR119ITGB3ITGAV
SCHEMBL8344058 0.81 GPR119 (0.42) GPR119MMP13ITGB3ITGAVITGA2B
SCHEMBL8346388 0.75 GPR119 (0.43) NPC1RAB9AGPR119DPP4ALDH1A1
SCHEMBL13855089 0.75 ITGB3 (0.56) NPC1RAB9AGPR119ITGB3ITGAV
SCHEMBL10154213 0.74 P2RX7 (0.36) NPC1RAB9AALDH1A1MAPTITGB3
SCHEMBL12892122 0.71 ITGB3 (0.45) NPC1RAB9AGPR119MMP13EED
SCHEMBL8345087 0.68 GPR119 (0.47) NPC1RAB9AGPR119MMP13ALDH1A1
SCHEMBL8030519 0.68 ITGB3 (0.44) GPR119MMP13ITGB3ITGAVITGA2B
SCHEMBL13591240 0.66 ALDH1A1 (0.51) NPC1RAB9AGPR119ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539739-B1 PIPERIDINYL COMPOUNDS THAT SELECTIVELY BIND INTEGRINS JANSSEN PHARMACEUTICA NV (BE) 2010-11-24 EP disclosed
WO-2004020435-A1 PIPERIDINYL COMPOUNDS THAT SELECTIVELY BIND INTEGRINS JANSSEN PHARMACEUTICA N.V. (BE) 2004-03-11 WO disclosed