SCHEMBL8347203

SCHEMBL8347203

O=NC(=O)C1(c2ccc(F)cc2)CCN(Cc2ccccc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 7/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
OPRL1 P41146 1/20 0.48
CCR3 P51677 1/20 0.47
POLB P06746 1/20 0.47
CYP2D6 P10635 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460365 0.91 OPRL1 (0.57) MEN1KMT2AOPRL1CCR3POLB
SCHEMBL8349645 0.89 CCR3 (0.61) MEN1KMT2AOPRL1CCR3POLB
Hydrochloric Acid SCHEMBL8347459 0.88 ALDH1A1 (0.45) CACNA1GMEN1KMT2APOLBCYP2D6
SCHEMBL8347345 0.88 LMNA (0.52) MEN1KMT2AOPRL1CCR3POLB
SCHEMBL8349949 0.87 POLB (0.55) OPRL1POLBMAPK1
SCHEMBL2702170 0.85 ALDH1A1 (0.55) CACNA1GMEN1KMT2AOPRL1CCR3
SCHEMBL373427 0.84 SLC6A12 (0.53) CACNA1GMEN1KMT2ACYP2D6MAPK1
SCHEMBL8347214 0.81 CACNA1G (0.48) CACNA1GMEN1KMT2AOPRL1CCR3
SCHEMBL10924212 0.81 SLC6A12 (0.53) MEN1KMT2AOPRL1POLBCYP2D6
SCHEMBL7463193 0.78 OPRL1 (0.46) MEN1KMT2AOPRL1CCR3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5861416-A TREATMENT OF ASTHMA OR COUGH MERRELL PHARMACEUTICALS INC. (US) 1999-01-19 US disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed
US-5661160-A ADMINISTERING AN ANTITUSSIVE AGENT FOR TREATING COUGH; TACHYKININ ANTAGONISM, SUBSTANCE P AND NEUROKININ A ANTAGONISM MERRELL PHARMACEUTICALS INC. (US) 1997-08-26 US disclosed
US-5648366-A TACHYKININ ANTAGONISTS USEFUL IN TREATING ASTHMA MERRELL PHARMACEUTICALS INC. (US) 1997-07-15 US disclosed
US-5635510-A TACHYKININ (ESPECIALLY SUBSTANCE P AND NEUROKININ A) ANTAGONISTS; ANTIINFLAMMATORY AGENTS, ANALGESICS; NERVOUS SYSTEM DISORDERS; BRONCHODILATOR AGENTS MERRELL PHARMACEUTICALS INC. (US) 1997-06-03 US disclosed