SCHEMBL8348015

SCHEMBL8348015

Cc1ccccc1NC(=O)C(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.52
PDK2 Q15119 1/20 0.52
PDK3 Q15120 1/20 0.52
PDK4 Q16654 1/20 0.52
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
HPGD P15428 4/20 0.47
ALDH1A1 P00352 3/20 0.47
POLB P06746 3/20 0.44
LMNA P02545 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
ALOX12 P18054 1/20 0.42
EPHX1 P07099 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
HSD17B10 Q99714 1/20 0.41
DDX3X O00571 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38661613 0.85 GAA (0.48) PDK1PDK2PDK3PDK4NPC1
SCHEMBL1534089 0.84 NPC1 (0.58) PDK1PDK2PDK3PDK4NPC1
SCHEMBL38664167 0.84 HDAC1 (0.47) PDK1PDK2PDK3PDK4NPC1
SCHEMBL6824411 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4NPC1
SCHEMBL13497754 0.82 LMNA (0.40) PDK1PDK2PDK3PDK4ALDH1A1
SCHEMBL27428457 0.80 PDK1 (0.49) PDK1PDK2PDK3PDK4NPC1
SCHEMBL11245698 0.78 PDK1 (0.61) PDK1PDK2PDK3PDK4NPC1
O-Tolylamine SCHEMBL19586028 0.77 NPC1 (0.49) PDK1PDK2PDK3PDK4NPC1
SCHEMBL292651 0.77 MAPT (0.43) PDK1PDK2PDK3PDK4NPC1
SCHEMBL397003 0.76 PDK1 (0.67) PDK1PDK2PDK3PDK4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004022534-A1 ARYLGLYCINE DERIVATIVES FOR USE AS GLYCINE TRANSPORT INHIBITORS NPS ALLELIX CORP. (CA) 2004-03-18 WO disclosed