SCHEMBL8348202

SCHEMBL8348202

O=C(N[C@@H](Cc1ccc(O)cc1)C(=O)N1CC[C@@H]2[C@H]1C(=O)CN2C(=O)c1ccccc1)c1cccc2cccnc12

nearest known ligand 0.51

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.51
CTSS P25774 2/20 0.42
CTSL P07711 1/20 0.42
HCRTR1 O43613 13/20 0.41
HCRTR2 O43614 10/20 0.41
ACE P12821 1/20 0.38
ACE2 Q9BYF1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8347622 0.88 CTSK (0.55) CTSKCTSSCTSLACEACE2
SCHEMBL5941507 0.86 CTSK (0.67) CTSKCTSSCTSLACEACE2
SCHEMBL5941511 0.86 CTSK (0.67) CTSKCTSSCTSLACEACE2
SCHEMBL6209627 0.85 CHRNB2 (0.42) CTSKCTSSCTSLHCRTR1HCRTR2
SCHEMBL4217173 0.84 CTSK (0.57) CTSKCTSSCTSLACEACE2
SCHEMBL4217170 0.84 CTSK (0.57) CTSKCTSSCTSLACEACE2
SCHEMBL5942475 0.84 CTSK (0.57) CTSKCTSSCTSLACEACE2
SCHEMBL13909143 0.84 CTSK (0.52) CTSKCTSSCTSL
SCHEMBL8349386 0.84 CTSK (0.52) CTSKCTSSCTSLACEACE2
SCHEMBL6210598 0.84 CTSL (0.45) CTSKCTSSCTSLACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed