SCHEMBL6209627

SCHEMBL6209627

O=C(NC(Cc1ccc(O)cc1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1)c1cccc2cccnc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
CTSK P43235 3/20 0.39
CTSS P25774 3/20 0.39
CTSL P07711 2/20 0.39
CYP51A1 Q16850 1/20 0.36
PREP P48147 1/20 0.36
ACE P12821 2/20 0.35
HCRTR1 O43613 4/20 0.35
HCRTR2 O43614 4/20 0.35
ACE2 Q9BYF1 1/20 0.35
GPR132 Q9UNW8 4/20 0.34
CMKLR2 P46091 1/20 0.34
CMKLR1 Q99788 1/20 0.34
CAPN1 P07384 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CTSB P07858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6212077 0.91 CTSL (0.39) CTSKCTSSCTSLCYP51A1PREP
SCHEMBL8348202 0.85 CTSK (0.51) CTSKCTSSCTSLACEHCRTR1
SCHEMBL4046533 0.83 MAPK1 (0.36) CTSKCTSSCYP51A1ACEACE2
SCHEMBL4043376 0.83 CTSK (0.56) CHRNB2CHRNA4CTSKCTSSACE
SCHEMBL4049549 0.80 GPR132 (0.38) CTSKCTSSACEACE2GPR132
SCHEMBL4043491 0.80 DPP4 (0.48)
SCHEMBL6210816 0.79 CTSL (0.43) CTSKCTSSCTSLHCRTR1HCRTR2
SCHEMBL6209046 0.79 CTSK (0.47) CTSKCTSSCTSLCYP51A1ACE
SCHEMBL4046323 0.78 CTSK (0.54) CTSKCTSSCTSLCYP51A1ACE
SCHEMBL6210598 0.77 CTSL (0.45) CTSKCTSSCTSLPREPACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-A1 BIOLOGICALLY ACTIVE COMPOUNDS Amura Therapeutics Limited (GB) 2005-06-29 EP disclosed
WO-2004007501-A1 BIOLOGICALLY ACTIVE COMPOUNDS AMURA THERAPEUTICS LIMITED (GB) 2004-01-22 WO disclosed