SCHEMBL8350468

SCHEMBL8350468

NC(=O)Nc1ccc2nc(N)nc(N)c2c1

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.54
MEN1 O00255 1/20 0.48
MMP1 P03956 1/20 0.48
MMP9 P14780 1/20 0.48
ALOX15 P16050 1/20 0.48
BLM P54132 1/20 0.48
GNG2 P59768 1/20 0.48
GNB1 P62873 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6094062 0.84 DHFR (0.53) DHFR
SCHEMBL28854429 0.76 GNG2 (0.81) MEN1MMP1MMP9ALOX15BLM
SCHEMBL4357022 0.76 MAP4K4 (0.54) DHFRMEN1KMT2A
SCHEMBL8222070 0.76 DHFR (0.57) DHFR
SCHEMBL10479133 0.75 MAOB (0.53) MEN1KMT2A
SCHEMBL6095892 0.75 ULK1 (0.61) DHFR
SCHEMBL29010947 0.74 DHFR (0.59) DHFR
SCHEMBL6004946 0.74 DHFR (0.69) DHFR
SCHEMBL30795245 0.74 DHFR (0.69) DHFR
SCHEMBL4753528 0.73 TDP1 (0.51) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999025327-A2 SMALL MOLECULE INTERVENTION IN HIV-1 REPLICATION WARNER-LAMBERT COMPANY (US) 1999-05-27 WO claimed
WO-1999025327-A2 SMALL MOLECULE INTERVENTION IN HIV-1 REPLICATION WARNER-LAMBERT COMPANY (US) 1999-05-27 WO disclosed