SCHEMBL8352011

SCHEMBL8352011

CC(C)C[C@H](N[C@@H](c1ccc(Cl)nc1)C(F)(F)F)C(=O)NC1(N)CC1

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSL P07711 15/20 0.52
CTSK P43235 9/20 0.49
CTSS P25774 9/20 0.47
CTSB P07858 8/20 0.47
GRN P28799 1/20 0.44
SORT1 Q99523 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2155255 0.86 CTSL (0.72) CTSLCTSKCTSSCTSB
SCHEMBL2155758 0.82 GRN (0.64) CTSLCTSKCTSSCTSBGRN
SCHEMBL12327770 0.82 CTSL (0.50) CTSLCTSKCTSSCTSB
SCHEMBL8293572 0.77 CTSK (0.76) CTSLCTSKCTSSCTSB
SCHEMBL8294942 0.76 CTSL (0.61) CTSLCTSKCTSSCTSB
SCHEMBL8294127 0.76 CTSL (0.61) CTSLCTSKCTSSCTSB
SCHEMBL14672982 0.76 CTSL (0.53) CTSLCTSKCTSSCTSB
SCHEMBL8293576 0.74 CTSL (0.54) CTSLCTSKCTSSCTSB
SCHEMBL2155322 0.73 GRN (0.41) CTSLCTSKCTSSCTSBGRN
SCHEMBL8236603 0.72 CTSL (0.54) CTSLCTSKCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1482924-B1 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA LTD (CA) 2008-05-21 EP disclosed
WO-2003075836-A2 CATHEPSIN CYSTEINE PROTEASE INHIBITORS MERCK FROSST CANADA & CO. (CA) 2003-09-18 WO disclosed