SCHEMBL8352109

SCHEMBL8352109

O=C(O)c1cn2ccc(CN[PH](=O)O)nc2n1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
KDM4E B2RXH2 2/20 0.30
HPGD P15428 2/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
MAPT P10636 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8346739 0.74 PGK1 (0.44) PTGS1PTGS2KDM4EHPGDALDH1A1
SCHEMBL8351974 0.74 PDCD1 (0.34) PTGS1PTGS2KDM4EHPGDALDH1A1
SCHEMBL8346722 0.70 KDM4E (0.33) KDM4E
SCHEMBL23571486 0.69 PTGS1 (0.47) PTGS1PTGS2KDM4EHPGDALDH1A1
SCHEMBL22777781 0.64 DHODH (0.49) PTGS1PTGS2KDM4EHPGDALDH1A1
SCHEMBL8346853 0.63 KDM4E (0.31) KDM4E
SCHEMBL8347708 0.62 VNN1 (0.32)
SCHEMBL570407 0.61 ALDH1A1 (0.61) PTGS1PTGS2KDM4EHPGDALDH1A1
SCHEMBL8348909 0.59 KDM4E (0.35) PTGS1PTGS2KDM4EALDH1A1MAPT
SCHEMBL8349224 0.59 EED (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5958904-A Phosphonomethyl-imidazo 1,2-A! pyrimidine-2-carboxylic acid compounds for treatment of neurotoxic injury G.D. SEARLE & CO. (US) 1999-09-28 US disclosed