SCHEMBL8355196

SCHEMBL8355196

CCCn1c(=O)[nH]c2ncn(C)c2c1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.64
BLM P54132 2/20 0.64
PMP22 Q01453 2/20 0.64
ALDH1A1 P00352 1/20 0.64
LMNA P02545 1/20 0.64
MAPT P10636 1/20 0.64
TSHR P16473 1/20 0.64
ADORA2A P29274 11/20 0.60
PDE4A P27815 10/20 0.60
PDE4B Q07343 10/20 0.60
PDE4C Q08493 10/20 0.60
PDE4D Q08499 10/20 0.60
ADORA2B P29275 4/20 0.56
CYP1A2 P05177 1/20 0.56
HSD17B10 Q99714 1/20 0.56
ADORA3 P0DMS8 2/20 0.56
GDA Q9Y2T3 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26925735 0.89 CYP3A4 (0.66) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL7403404 0.80 ALDH1A1 (0.57) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL8061720 0.79 LMNA (0.54) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL7101360 0.79 BLM (0.54) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL11442354 0.79 BLM (0.54) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL9844553 0.79 PDE4A (0.56) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL6344281 0.78 LMNA (0.52) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL6344284 0.78 LMNA (0.52) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL6357569 0.78 LMNA (0.52) CYP3A4BLMPMP22ALDH1A1LMNA
SCHEMBL12080148 0.78 ADORA2A (0.47) CYP3A4BLMPMP22ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031101-A1 ADENOSINE RECEPTOR ANTAGONISTS WITH IMPROVED BIOACTIVITY UNIVERSITY OF SOUTH FLORIDA (US) 1999-06-24 WO disclosed