SCHEMBL9844553

SCHEMBL9844553

CCCn1cnc2[nH]c(=O)n(CC)c(=O)c21

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.56
ADORA2A P29274 6/20 0.56
PDE4B Q07343 6/20 0.56
PDE4C Q08493 6/20 0.56
PDE4D Q08499 6/20 0.56
CNOT7 Q9UIV1 4/20 0.52
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ADORA2B P29275 2/20 0.47
ADORA3 P0DMS8 1/20 0.47
BRD4 O60885 1/20 0.46
BRD2 P25440 1/20 0.46
BRD3 Q15059 1/20 0.46
BRDT Q58F21 1/20 0.46
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
MAPT P10636 1/20 0.45
TSHR P16473 1/20 0.45
BLM P54132 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10812168 0.89 PDE4A (0.53) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL26925735 0.83 CYP3A4 (0.66) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL13861874 0.81 CNOT7 (0.70) ADORA2ACNOT7ALDH1A1MEN1KMT2A
SCHEMBL9293981 0.79 CNOT7 (0.47) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8355196 0.79 CYP3A4 (0.64) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9293978 0.78 CNOT7 (0.43) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL13217674 0.77 ALDH1A1 (0.66) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7464482 0.77 PDE4A (0.86) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL27461932 0.77 PDE4A (0.49) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL8660274 0.76 CNOT7 (0.49) PDE4AADORA2APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413278-A2 Use of xanthine derivatives against peptic ulcers HOECHST JAPAN LIMITED (JP) 1991-02-20 EP disclosed