SCHEMBL8358995

SCHEMBL8358995

CCCn1c(=O)[nH]c(=O)c2ncn(COC(=O)C(C)(C)C)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 7/20 0.44
PDE4B Q07343 7/20 0.44
PDE4C Q08493 7/20 0.44
PDE4D Q08499 7/20 0.44
ADORA2A P29274 6/20 0.44
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TK1 P04183 1/20 0.38
ADORA2B P29275 2/20 0.38
ADORA3 P0DMS8 1/20 0.38
HPGD P15428 1/20 0.38
ADORA1 P30542 1/20 0.38
BLM P54132 1/20 0.38
PDE3A Q14432 1/20 0.38
HSD17B10 Q99714 1/20 0.38
BRD4 O60885 1/20 0.37
BRD2 P25440 1/20 0.37
BRD3 Q15059 1/20 0.37
BRDT Q58F21 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4623458 0.80 PDE4A (0.63) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL6251096 0.77 PDE4A (0.64) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL3990425 0.75 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL8355211 0.74 PNP (0.44) MEN1KMT2AALDH1A1TK1BLM
SCHEMBL4626797 0.73 BRD4 (0.65) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL7672450 0.71 PNP (0.63) MEN1KMT2AALDH1A1TK1BLM
SCHEMBL16510025 0.68 POLB (0.42) KMT2AADORA2BPOLBGAANPSR1
SCHEMBL9200960 0.68 ALDH1A1 (0.51) ADORA2AALDH1A1TK1ADORA2BBLM
SCHEMBL5476039 0.68 TK1 (0.67) TK1HPGD
SCHEMBL5789121 0.68 KDM4E (0.55) PDE4APDE4BPDE4CPDE4DADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999031101-A1 ADENOSINE RECEPTOR ANTAGONISTS WITH IMPROVED BIOACTIVITY UNIVERSITY OF SOUTH FLORIDA (US) 1999-06-24 WO disclosed