Dimethyl Maleate

Dimethyl Maleate

SCHEMBL8359457

COC(=O)/C=C\C(=O)OC.CO[Si](CCCN)(OC)OC

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

KEAP1

The experimentally established mechanism targets of Dimethyl Maleate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 known ✓ Q14145 1/20 0.48
NFE2L2 Q16236 3/20 0.48
HCAR2 Q8TDS4 2/20 0.48
GFPT1 Q06210 1/20 0.40
PAOX Q6QHF9 2/20 0.33
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ATM Q13315 1/20 0.31
LMNA P02545 2/20 0.30
HTT P42858 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
RAB9A P51151 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
TYR P14679 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Dimethyl Fumarate SCHEMBL8359467 1.00 NFE2L2 (0.48) NFE2L2HCAR2KEAP1GFPT1PAOX
Bicarbonate SCHEMBL18662974 0.82 LMNA (0.37) PAOXALDH1A1LMNAMEN1KMT2A
Urea SCHEMBL27918835 0.82 PAOX (0.34) PAOXALDH1A1LMNAMEN1KMT2A
Acetone SCHEMBL2390270 0.82 PAOX (0.39) PAOXALDH1A1LMNAMEN1KMT2A
SCHEMBL4605785 0.80 ATM (0.61) HCAR2MAPTALDH1A1TDP1ATM
Acetic Acid SCHEMBL28413060 0.80 PAOX (0.38) PAOXALDH1A1LMNAMEN1KMT2A
Acetic Acid SCHEMBL5065362 0.80 PAOX (0.38) PAOXALDH1A1LMNAMEN1KMT2A
Acetic Acid SCHEMBL28413059 0.80 PAOX (0.38) PAOXALDH1A1LMNAMEN1KMT2A
Acetic Acid SCHEMBL3253044 0.80 PAOX (0.38) PAOXALDH1A1LMNAMEN1KMT2A
SCHEMBL7096198 0.80 ATM (0.50) NFE2L2HCAR2KEAP1GFPT1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6001946-A Curable silane-encapped compositions having improved performances WITCO CORPORATION (US) 1999-12-14 US disclosed