SCHEMBL8360277

SCHEMBL8360277

CCCCCCC(NC(=O)Cc1c(C)n(C(=O)c2ccccc2)c2ccc(OC)cc12)C(=O)N(CCCC)CCCC

nearest known ligand 0.59

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
TSHR P16473 1/20 0.59
NFKB1 P19838 1/20 0.59
HIF1A Q16665 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
PTGS2 P35354 14/20 0.59
PLA2G2A P14555 1/20 0.57
AKR1C3 P42330 1/20 0.53
AKR1C2 P52895 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8358919 0.94 LMNA (0.61) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8354810 0.93 LMNA (0.58) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8354816 0.92 LMNA (0.59) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8356800 0.89 LMNA (0.59) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8361046 0.88 PTGS2 (0.62) NPSR1PTGS2AKR1C3AKR1C2
SCHEMBL8360017 0.88 LMNA (0.62) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8360240 0.87 PTGS2 (0.60) NPSR1PTGS2AKR1C3AKR1C2
SCHEMBL8354773 0.87 PTGS2 (0.71) PTGS2
SCHEMBL8356449 0.86 LMNA (0.50) LMNACYP1A2CYP2D6CYP2C9TSHR
SCHEMBL8356332 0.86 PTGS2 (0.59) PTGS2AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5877202-A Indole derivatives useful to treat estrogen-related neoplasms and disorders AVENTISUB II INC. 1999-03-02 US disclosed