SCHEMBL8364438

SCHEMBL8364438

Cn1c(=O)cc(CCO)c2cc(F)ccc21

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.43
BRD4 O60885 6/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HPGD P15428 2/20 0.41
ATM Q13315 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
XIAP P98170 1/20 0.39
ICMT O60725 2/20 0.38
HSD17B10 Q99714 2/20 0.38
HCRTR1 O43613 1/20 0.38
NQO2 P16083 1/20 0.37
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8366153 0.85 THRB (0.43) THRBBRD4HTTKDM4EALDH1A1
SCHEMBL8366307 0.82 ALDH1A1 (0.47) THRBHTTALDH1A1HPGDRXFP1
SCHEMBL15565909 0.82 THRB (0.42) THRBBRD4HTTKDM4EALDH1A1
SCHEMBL8367148 0.81 AKR1C3 (0.49) THRBBRD4HTTKDM4EALDH1A1
SCHEMBL9153374 0.80 KDM4E (0.56) BRD4HTTKDM4EALDH1A1HPGD
SCHEMBL8366314 0.79 BRD1 (0.42) BRD4HSD17B10
SCHEMBL8366324 0.78 THRB (0.47) THRBBRD4HTTKDM4EALDH1A1
SCHEMBL21614279 0.77 KDM4E (0.50) KDM4EALDH1A1MEN1KMT2ARXFP1
SCHEMBL31563337 0.77 KDM4E (0.41) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL13440436 0.76 KDM4E (0.50) THRBBRD4KDM4EALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850235-B1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SANOFI SYNTHELABO (FR) 1999-12-01 EP disclosed
US-5958924-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS, RESTENOSIS, ANTICOALUGANTS, RESPIRATORY SYSTEM DISORDERS SYNTHELABO (FR) 1999-09-28 US disclosed