SCHEMBL8366307

SCHEMBL8366307

Cn1c(=O)cc(CCO)c2cc(Cl)ccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RXFP1 Q9HBX9 5/20 0.46
CNR1 P21554 1/20 0.44
TP53 P04637 1/20 0.43
CYP2C9 P11712 2/20 0.43
MAPT P10636 2/20 0.43
KCNH2 Q12809 2/20 0.42
THRB P10828 1/20 0.41
GAA P10253 1/20 0.41
ALOX15 P16050 2/20 0.40
TSHR P16473 2/20 0.40
MAPK8 P45983 2/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8369444 0.87 ALDH1A1 (0.45) ALDH1A1HTTSMN1; SMN2RXFP1CNR1
SCHEMBL8364438 0.82 THRB (0.43) ALDH1A1HTTRXFP1KCNH2THRB
SCHEMBL8364439 0.81 ALDH1A1 (0.49) ALDH1A1HTTSMN1; SMN2RXFP1TP53
SCHEMBL9153374 0.80 KDM4E (0.56) ALDH1A1HTTSMN1; SMN2MAPTGAA
SCHEMBL8366314 0.79 BRD1 (0.42) MAPTHSD17B10
SCHEMBL6242735 0.77 CDK2 (0.47) RXFP1KCNH2
SCHEMBL21979134 0.74 NQO2 (0.61) ALDH1A1HTTSMN1; SMN2RXFP1TP53
SCHEMBL5780369 0.72 CNR1 (0.57) SMN1; SMN2RXFP1CNR1MAPT
SCHEMBL24095575 0.72 HSD17B10 (0.69) RXFP1MAPTALOX15TSHRLMNA
SCHEMBL8366153 0.71 THRB (0.43) ALDH1A1HTTSMN1; SMN2RXFP1CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0850235-B1 QUINOLEIN-2(1H)-ONE DERIVATIVES AS SEROTONIN ANTAGONISTS SANOFI SYNTHELABO (FR) 1999-12-01 EP disclosed
US-5958924-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS, RESTENOSIS, ANTICOALUGANTS, RESPIRATORY SYSTEM DISORDERS SYNTHELABO (FR) 1999-09-28 US disclosed