SCHEMBL8366149

SCHEMBL8366149

CCOC(=O)CC(=O)Cc1cccc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.56
TDP1 Q9NUW8 2/20 0.53
ATM Q13315 1/20 0.52
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
L3MBTL1 Q9Y468 3/20 0.51
KDM4E B2RXH2 1/20 0.51
APOBEC3A P31941 1/20 0.51
APOBEC3G Q9HC16 1/20 0.51
SIRT5 Q9NXA8 1/20 0.49
LMNA P02545 1/20 0.48
PKM P14618 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
MAPK10 P53779 1/20 0.47
CDC25B P30305 2/20 0.47
CDC25A P30304 1/20 0.47
CDC25C P30307 1/20 0.47
MTNR1A P48039 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30070191 1.00 KMT2A (0.56) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL29729685 0.88 KMT2A (0.62) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL845701 0.88 KMT2A (0.62) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL30716618 0.86 KMT2A (0.54) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL20897263 0.86 KMT2A (0.54) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL8402588 0.81 NLRP3 (0.48) KMT2AALDH1A1PKMSMN1; SMN2CYP4F2
SCHEMBL31751033 0.81 NLRP3 (0.48) KMT2AALDH1A1PKMSMN1; SMN2CYP4F2
SCHEMBL10820834 0.80 TDP1 (0.61) KMT2ATDP1ATMALDH1A1HPGD
SCHEMBL28332298 0.79 KMT2A (0.53) KMT2ATDP1ALDH1A1HPGDL3MBTL1
SCHEMBL11313603 0.79 MTNR1A (0.45) KMT2AALDH1A1HPGDL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230131899-A1 INHIBITORS OF MICROBIALLY INDUCED AMYLOID AXIAL THERAPEUTICS, INC. (US) 2023-04-27 US disclosed
US-20230131899-A1 INHIBITORS OF MICROBIALLY INDUCED AMYLOID AXIAL THERAPEUTICS, INC. (US) 2023-04-27 US disclosed
US-20230131899-A1 INHIBITORS OF MICROBIALLY INDUCED AMYLOID AXIAL THERAPEUTICS, INC. (US) 2023-04-27 US disclosed
EP-4087560-A2 INHIBITORS OF MICROBIALLY INDUCED AMYLOID Axial Therapeutics, Inc. (US) 2022-11-16 EP disclosed
CN-102134223-A Preparation and application of novel chiral 3,4-dihydro-2-alkoxyl-6-benzyl-4-oxopyrimidine (S-DABO) human immunodeficiency virus (HIV)-1 reverse transcriptase inhibitor UNIV CAPITAL MEDICAL 2011-07-27 CN disclosed
US-5929067-A N-ACYLATING AMINE DERIVATIVE OF CAPROLACTAM COMPOUND WITH A CARBOXYLIC ACID OR DERIVATIVES TO FORM AMIDE DERIVATIVE OF CAPROLACTAM COMPOUND NOVARTIS AG (CH) 1999-07-27 US disclosed
EP-0810991-B1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1999-04-14 EP disclosed
EP-0810991-A1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS Novartis AG (CH) 1997-12-10 EP disclosed
WO-1996026183-A1 1-ARYL-2-ACYLAMINO-ETHANE COMPOUNDS AND THEIR USE AS NEUROKININ ESPECIALLY NEUROKININ 1 ANTAGONISTS NOVARTIS AG (CH) 1996-08-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230131899-A1 INHIBITORS OF MICROBIALLY INDUCED AMYLOID SNCA, PARK7, PRNP KMT2A 4786/4885TDP1 452/4885ATM 3731/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.