SCHEMBL8364439

SCHEMBL8364439

Cn1c(=O)cc(CC(=O)O)c2cc(Cl)ccc21

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MAPT P10636 2/20 0.48
KDM4E B2RXH2 1/20 0.48
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
RXFP1 Q9HBX9 5/20 0.47
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
GAA P10253 1/20 0.45
TP53 P04637 1/20 0.45
AKR1C3 P42330 2/20 0.44
AKR1C2 P52895 2/20 0.44
AKR1C4 P17516 1/20 0.44
PTGS1 P23219 1/20 0.44
OXER1 Q8TDS5 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9766045 0.84 MEN1 (0.51) ALDH1A1SMN1; SMN2MAPTKDM4EHPGD
SCHEMBL8367148 0.83 AKR1C3 (0.49) ALDH1A1HTTMAPTKDM4EHPGD
SCHEMBL8457832 0.83 KDM4E (0.48) ALDH1A1SMN1; SMN2MAPTKDM4EHPGD
SCHEMBL8366307 0.81 ALDH1A1 (0.47) ALDH1A1HTTSMN1; SMN2MAPTHPGD
SCHEMBL9157244 0.81 KDM4E (0.56) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL9156302 0.81 KDM4E (0.46) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL8366206 0.81 KDM4E (0.55) ALDH1A1SMN1; SMN2MAPTKDM4EHPGD
SCHEMBL8366369 0.80 ALDH1A1 (0.44) ALDH1A1MAPTKDM4EHPGDHSD17B10
SCHEMBL6242130 0.79 KMT2A (0.52) ALDH1A1HTTMAPTKDM4EHPGD
SCHEMBL8369444 0.79 ALDH1A1 (0.45) ALDH1A1HTTSMN1; SMN2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1094490-C Quinolin-2 (1H) -one derivatives as serotonin antagonists SANOFI SYNTHELABO (FR) 2002-11-20 CN disclosed
US-5958924-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS, RESTENOSIS, ANTICOALUGANTS, RESPIRATORY SYSTEM DISORDERS SYNTHELABO (FR) 1999-09-28 US disclosed
CN-1202168-A Quinolein-2(1H)-one derivatives as serotonin antagonists SYNTHELABO (FR) 1998-12-16 CN disclosed