SCHEMBL8366338

SCHEMBL8366338

Fc1cccc([CH]Cc2cccc(F)c2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 6/20 0.54
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
PKM P14618 1/20 0.48
MAPK1 P28482 1/20 0.48
THPO P40225 1/20 0.48
CHRM5 P08912 1/20 0.48
GRM5 P41594 1/20 0.48
BLM P54132 1/20 0.48
PMP22 Q01453 1/20 0.48
TAAR1 Q96RJ0 3/20 0.47
IDO1 P14902 2/20 0.46
AGXT P21549 2/20 0.46
PTGS1 P23219 2/20 0.43
PTGS2 P35354 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840811 0.90 NFE2L2 (0.52) NFE2L2MAOAMAOBNPC1RAB9A
SCHEMBL5941183 0.86 NFE2L2 (0.50) NFE2L2MAOAMAOBNPC1RAB9A
SCHEMBL154188 0.86 NFE2L2 (0.55) NFE2L2MAOAMAOBNPC1RAB9A
SCHEMBL9187662 0.82 NFE2L2 (0.59) NFE2L2MAOAMAOBNPC1RAB9A
SCHEMBL28126527 0.81 NFE2L2 (0.61) NFE2L2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL7817239 0.80 MAOB (0.60) MAOAMAOBPKM
SCHEMBL8325508 0.77 NFE2L2 (0.55) NFE2L2MAOAMAOBNPC1RAB9A
SCHEMBL23457236 0.77 NFE2L2 (0.60) NFE2L2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL16618839 0.77 NFE2L2 (0.60) NFE2L2NPC1RAB9ACYP1A2CYP3A4
SCHEMBL167999 0.77 TAAR1 (0.52) NFE2L2MAOAMAOBNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929217-A4 SORDARIN DERIVATIVES MERCK & CO INC (US) 1999-12-15 EP disclosed
EP-0929217-A1 SORDARIN DERIVATIVES Merck & Co., Inc. (US) 1999-07-21 EP disclosed
WO-1998015178-A1 SORDARIN DERIVATIVES MERCK & CO., INC. (US) 1998-04-16 WO disclosed